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1-{2-[(4-chlorophenyl)amino]-2-oxoethyl}-N-(1-isopropylpiperidin-4-yl)-1H-indole-2-carboxamide

Development stage: Preclinical
Modality: Small Molecules

Overview

This compound is a synthetic small molecule belonging to the indolecarboxamide class, specifically an indole derivative. It is identified as an experimental agent and has been studied primarily as a potent inhibitor of coagulation factor X (F10), a serine protease involved in the blood coagulation cascade. The compound binds to factor X with high affinity (Ki ≈ 3 nM), suggesting potential anticoagulant activity. There are no approved therapeutic indications or marketed formulations for this molecule, and it remains at the research stage[6][5][9].

Other names: 1-{[(4-chlorophenyl)carbamoyl]methyl}-N-[1-(propan-2-yl)piperidin-4-yl]-1H-indole-2-carboxamide1-(2-((4-chlorophenyl)amino)-2-oxoethyl)-N-(1-isopropylpiperidin–4-YL)-1H-indole–2-carboxamide

Targets

F10 (Factor Xa)

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